Antigen Information
General Information of This Antigen
| Antigen ID | TAR0GLSWQ |
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|---|---|---|---|---|---|---|
| Antigen Name | CD276 antigen (CD276) |
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| Gene Name | CD276 |
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| Gene ID | ||||||
| Synonym | B7H3; PSEC0249; UNQ309; PRO352; 4Ig-B7-H3;B7 homolog 3;Costimulatory molecule;CD_antigen=CD276 |
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| Sequence |
MLRRRGSPGMGVHVGAALGALWFCLTGALEVQVPEDPVVALVGTDATLCCSFSPEPGFSL
AQLNLIWQLTDTKQLVHSFAEGQDQGSAYANRTALFPDLLAQGNASLRLQRVRVADEGSF TCFVSIRDFGSAAVSLQVAAPYSKPSMTLEPNKDLRPGDTVTITCSSYQGYPEAEVFWQD GQGVPLTGNVTTSQMANEQGLFDVHSILRVVLGANGTYSCLVRNPVLQQDAHSSVTITPQ RSPTGAVEVQVPEDPVVALVGTDATLRCSFSPEPGFSLAQLNLIWQLTDTKQLVHSFTEG RDQGSAYANRTALFPDLLAQGNASLRLQRVRVADEGSFTCFVSIRDFGSAAVSLQVAAPY SKPSMTLEPNKDLRPGDTVTITCSSYRGYPEAEVFWQDGQGVPLTGNVTTSQMANEQGLF DVHSVLRVVLGANGTYSCLVRNPVLQQDAHGSVTITGQPMTFPPEALWVTVGLSVCLIAL LVALAFVCWRKIKQSCEEENAGAEDQDGEGEGSKTALQPLKHSDSKEDDGQEIA Click to Show/Hide
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| Family | HIV-1 env protein family |
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| Function |
May participate in the regulation of T-cell-mediated immune response. May play a protective role in tumor cells by inhibiting natural-killer mediated cell lysis as well as a role of marker for detection of neuroblastoma cells. May be involved in the development of acute and chronic transplant rejection and in the regulation of lymphocytic activity at mucosal surfaces. Could also play a key role in providing the placenta and fetus with a suitable immunological environment throughout pregnancy. Both isoform 1 and isoform 2 appear to be redundant in their ability to modulate CD4 T-cell responses. Isoform 2 is shown to enhance the induction of cytotoxic T-cells and selectively stimulates interferon gamma production in the presence of T-cell receptor signaling.
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| Uniprot Entry | ||||||
| HGNC ID | ||||||
| KEGG ID | ||||||
Each Antibody-drug Conjuate AND It's Component Related to This Antigen
Full List of The ADC Related to This Antigen
1D1-01
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
1D1-01-ADC-Tb1-1 |
1D1-01-ADC-Tb1-1 payload |
Undisclosed |
1D1-01-ADC-Tb1-1 linker |
[1] | |
1D1-01-ADC-Tb1-2 |
1D1-01-ADC-Tb1-2 payload |
Undisclosed |
1D1-01-ADC-Tb1-2 linker |
[1] | |
1D1-01-ADC-Tb1-3 |
1D1-01-ADC-Tb1-3 payload |
Undisclosed |
1D1-01-ADC-Tb1-3 linker |
[1] | |
1D1-01-ADC-Tb1-4 |
1D1-01-ADC-Tb1-4 payload |
Undisclosed |
1D1-01-ADC-Tb1-4 linker |
[1] | |
1D1-01-ADC-Tb1-5 |
1D1-01-ADC-Tb1-5 payload |
Undisclosed |
1D1-01-ADC-Tb1-5 linker |
[1] | |
1D1-01-ADC-Tb1-6 |
1D1-01-ADC-Tb1-6 payload |
Undisclosed |
1D1-01-ADC-Tb1-6 linker |
[1] | |
1D1-01-ADC-Tb1-7 |
1D1-01-ADC-Tb1-7 payload |
Undisclosed |
1D1-01-ADC-Tb1-7 linker |
[1] | |
1D1-01-ADC-Tb1-8 |
1D1-01-ADC-Tb1-8 payload |
Undisclosed |
1D1-01-ADC-Tb1-8 linker |
[1] | |
1D1-01-ADC-Tb1-9 |
1D1-01-ADC-Tb1-9 payload |
Undisclosed |
1D1-01-ADC-Tb1-9 linker |
[1] | |
1D1-01-ADC-Tb1-10 |
1D1-01-ADC-Tb1-10 payload |
Undisclosed |
1D1-01-ADC-Tb1-10 linker |
[1] | |
1D1-01-ADC-Tb1-11 |
1D1-01-ADC-Tb1-11 payload |
Undisclosed |
1D1-01-ADC-Tb1-11 linker |
[1] | |
1D1-01-ADC-Tb1-12 |
1D1-01-ADC-Tb1-12 payload |
Undisclosed |
1D1-01-ADC-Tb1-12 linker |
[1] | |
1D1-01-ADC-Tb1-13 |
1D1-01-ADC-Tb1-13 payload |
Undisclosed |
1D1-01-ADC-Tb1-13 linker |
[1] | |
1D1-01-ADC-Tb1-14 |
1D1-01-ADC-Tb1-14 payload |
Undisclosed |
1D1-01-ADC-Tb1-14 linker |
[1] | |
1D1-01-ADC-Tb1-15 |
1D1-01-ADC-Tb1-15 payload |
Undisclosed |
1D1-01-ADC-Tb1-15 linker |
[1] | |
1D1-01-ADC-Tb1-16 |
1D1-01-ADC-Tb1-16 payload |
Undisclosed |
1D1-01-ADC-Tb1-16 linker |
[1] | |
1D1-01-ADC-Tb1-17 |
1D1-01-ADC-Tb1-17 payload |
Undisclosed |
1D1-01-ADC-Tb1-17 linker |
[1] | |
1D1-01-ADC-Tb1-18 |
1D1-01-ADC-Tb1-18 payload |
Undisclosed |
1D1-01-ADC-Tb1-18 linker |
[1] | |
1D1-01-ADC-Tb1-19 |
1D1-01-ADC-Tb1-19 payload |
Undisclosed |
1D1-01-ADC-Tb1-19 linker |
[1] | |
1D1-01-ADC-Tb1-20 |
1D1-01-ADC-Tb1-20 payload |
Undisclosed |
1D1-01-ADC-Tb1-20 linker |
[1] | |
1D1-01-ADC-Tb1-21 |
1D1-01-ADC-Tb1-21 payload |
Undisclosed |
1D1-01-ADC-Tb1-21 linker |
[1] | |
1D1-01-ADC-Tb1-22 |
1D1-01-ADC-Tb1-22 payload |
Undisclosed |
1D1-01-ADC-Tb1-22 linker |
[1] | |
1D1-01-ADC-Tb1-23 |
1D1-01-ADC-Tb1-23 payload |
Undisclosed |
1D1-01-ADC-Tb1-23 linker |
[1] | |
1D1-01-ADC-Tb1-24 |
1D1-01-ADC-Tb1-24 payload |
Undisclosed |
1D1-01-ADC-Tb1-24 linker |
[1] | |
1D1-01-ADC-Tb1-25 |
1D1-01-ADC-Tb1-25 payload |
Undisclosed |
1D1-01-ADC-Tb1-25 linker |
[1] | |
1D1-01-ADC-Tb1-26 |
1D1-01-ADC-Tb1-26 payload |
Undisclosed |
1D1-01-ADC-Tb1-26 linker |
[1] |
1F9DS
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
WO2020063676A1 ADC-25 |
WO2020063676A1_ADC-25 payload |
Undisclosed |
WO2020063676A1_ADC-25 linker |
[2] | |
WO2020063676A1 ADC-26 |
WO2020063676A1_ADC-26 payload |
Undisclosed |
WO2020063676A1_ADC-26 linker |
[2] | |
WO2020063676A1 ADC-27 |
WO2020063676A1_ADC-27 payload |
Undisclosed |
WO2020063676A1_ADC-27 linker |
[2] | |
WO2020063676A1 ADC-28 |
WO2020063676A1_ADC-28 payload |
Undisclosed |
WO2020063676A1_ADC-28 linker |
[2] | |
WO2020063676A1 ADC-29 |
WO2020063676A1_ADC-29 payload |
Undisclosed |
WO2020063676A1_ADC-29 linker |
[2] | |
WO2020063676A1 ADC-30 |
WO2020063676A1_ADC-30 payload |
Undisclosed |
WO2020063676A1_ADC-30 linker |
[2] | |
WO2020063676A1 ADC-31 |
WO2020063676A1_ADC-31 payload |
Undisclosed |
WO2020063676A1_ADC-31 linker |
[2] |
7300
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
40285886 7300-LP1003 |
Camptothecin derivative 095 |
Undisclosed |
a polyethylene glycol-modified straight-link agent |
[3] | |
40285886 7300-LP2004 |
Camptothecin derivative 095 |
Undisclosed |
a polyethylene glycol-modified branched-link agent |
[3] | |
40285886 7300-LP3004 |
Camptothecin derivative 095 |
Undisclosed |
a PSar-modified branched-link agent |
[3] | |
40285886 7300-Deruxtecan |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[3] |
Anti-b7h3
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
WBP301088-X2 |
Topo1 inhibitor F |
DNA topoisomerase I (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[4] |
Anti-B7H3 mAb 2E3-02
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
B7H3-ADC-01 |
B7H3-ADC-01 payload |
Undisclosed |
B7H3-ADC-01 linker |
[1] | |
B7H3-ADC-02 |
B7H3-ADC-02 payload |
Undisclosed |
B7H3-ADC-02 linker |
[1] | |
B7H3-ADC-03 |
B7H3-ADC-03 payload |
Undisclosed |
B7H3-ADC-03 linker |
[1] | |
B7H3-ADC-04 (DAR8) |
B7H3-ADC-04 payload |
Undisclosed |
B7H3-ADC-04 linker |
[1] | |
B7H3-ADC-05 (DAR8) |
B7H3-ADC-05(DAR8) payload |
Undisclosed |
B7H3-ADC-05(DAR8) linker |
[1] | |
B7H3-ADC-05 (DAR4) |
B7H3-ADC-05(DAR8) payload |
Undisclosed |
B7H3-ADC-05(DAR4) linker |
[1] | |
B7H3-ADC-06 (DAR8) |
B7H3-ADC-06 payload |
Undisclosed |
B7H3-ADC-06 linker |
[1] | |
B7H3-ADC-07 (DAR8) |
B7H3-ADC-07(DAR8) payload |
Undisclosed |
B7H3-ADC-07(DAR8) linker |
[1] | |
B7H3-ADC-07 (DAR2) |
B7H3-ADC-07(DAR2) payload |
Undisclosed |
B7H3-ADC-07(DAR2) linker |
[1] | |
B7H3-ADC-07 (DAR4) |
B7H3-ADC-07(DAR4) payload |
Undisclosed |
B7H3-ADC-07(DAR4) linker |
[1] | |
B7H3-ADC-07 (DAR6) |
B7H3-ADC-07(DAR6) payload |
Undisclosed |
B7H3-ADC-07(DAR6) linker |
[1] | |
B7H3-ADC-08 (DAR8) |
B7H3-ADC-08(DAR8) payload |
Undisclosed |
B7H3-ADC-08(DAR8) linker |
[1] | |
B7H3-ADC-08 (DAR4) |
B7H3-ADC-08(DAR4) payload |
Undisclosed |
B7H3-ADC-08(DAR4) linker |
[1] | |
B7H3-ADC-09 (DAR8) |
B7H3-ADC-09 payload |
Undisclosed |
B7H3-ADC-09 linker |
[1] | |
B7H3-ADC-10 (DAR8) |
B7H3-ADC-10 payload |
Undisclosed |
B7H3-ADC-10 linker |
[1] | |
B7H3-ADC-11 (DAR8) |
B7H3-ADC-11 payload |
Undisclosed |
B7H3-ADC-11 linker |
[1] | |
B7H3-ADC-12 (DAR8) |
B7H3-ADC-12 payload |
Undisclosed |
B7H3-ADC-12 linker |
[1] | |
B7H3-ADC-13 (DAR8) |
B7H3-ADC-13 payload |
Undisclosed |
B7H3-ADC-13 linker |
[1] | |
B7H3-ADC-14 (DAR8) |
B7H3-ADC-14 payload |
Undisclosed |
B7H3-ADC-14 linker |
[1] | |
B7H3-ADC-15 (DAR8) |
B7H3-ADC-15(DAR8) payload |
Undisclosed |
B7H3-ADC-15(DAR8) linker |
[1] | |
B7H3-ADC-15 (DAR4) |
B7H3-ADC-15(DAR4) payload |
Undisclosed |
B7H3-ADC-15(DAR4) linker |
[1] | |
B7H3-ADC-16 (DAR8) |
B7H3-ADC-16 payload |
Undisclosed |
B7H3-ADC-16 linker |
[1] | |
B7H3-ADC-17 |
B7H3-ADC-17 payload |
Undisclosed |
B7H3-ADC-17 linker |
[1] | |
B7H3-ADC-18 (DAR8) |
B7H3-ADC-18 payload |
Undisclosed |
B7H3-ADC-18 linker |
[1] | |
B7H3-ADC-19 (DAR8) |
B7H3-ADC-19 payload |
Undisclosed |
B7H3-ADC-19 linker |
[1] | |
B7H3-ADC-20 (DAR8) |
B7H3-ADC-20 payload |
Undisclosed |
B7H3-ADC-20 linker |
[1] | |
B7H3-ADC-22 (DAR8) |
B7H3-ADC-22 payload |
Undisclosed |
B7H3-ADC-22 linker |
[1] | |
B7H3-ADC-23 (DAR8) |
B7H3-ADC-23 payload |
Undisclosed |
B7H3-ADC-23 linker |
[1] | |
B7H3-ADC-24 (DAR8) |
B7H3-ADC-24 payload |
Undisclosed |
B7H3-ADC-24 linker |
[1] | |
B7H3-ADC-25 (DAR8) |
B7H3-ADC-25 payload |
Undisclosed |
B7H3-ADC-25 linker |
[1] | |
B7H3-ADC-27 (DAR8) |
B7H3-ADC-27 payload |
Undisclosed |
B7H3-ADC-27 linker |
[1] | |
B7H3-ADC-28 (DAR8) |
B7H3-ADC-28 payload |
Undisclosed |
B7H3-ADC-28 linker |
[1] | |
B7H3-ADC-32 (DAR8) |
B7H3-ADC-32 payload |
Undisclosed |
B7H3-ADC-32 linker |
[1] | |
B7H3-ADC-33 (DAR8) |
B7H3-ADC-33(DAR8) payload |
Undisclosed |
B7H3-ADC-33(DAR8) linker |
[1] | |
B7H3-ADC-33 (DAR4) |
B7H3-ADC-33(DAR4) payload |
Undisclosed |
B7H3-ADC-33(DAR4) linker |
[1] | |
B7H3-ADC-001 |
DL014-payload; DL003-payload |
Undisclosed |
DL014-Linker; DL003-Linker |
[5] | |
B7H3-ADC-002 |
DL014-payload; DL003-payload |
Undisclosed |
DL014-Linker; DL003-Linker |
[5] | |
B7H3-ADC-003 |
DL014-payload; DL003-payload |
Undisclosed |
DL014-Linker; DL003-Linker |
[5] |
Anti-CD276 mAb
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
Anti-CD276 mAb-MMAF |
Monomethyl auristatin F |
Microtubule (MT) |
Undisclosed |
[6] |
Anti-CD276 mAb h1702DS
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
WO2020063673A1 ADC-1 |
WO2020063673A1_ADC-1 payload |
Undisclosed |
WO2020063673A1_ADC-1 linker |
[7] | |
WO2020063673A1 ADC-2 |
WO2020063673A1_ADC-2 payload |
Undisclosed |
WO2020063673A1_ADC-2 linker |
[7] | |
WO2020063673A1 ADC-3 |
WO2020063673A1_ADC-3 payload |
Undisclosed |
WO2020063673A1_ADC-3 linker |
[7] | |
WO2020063673A1 ADC-4 |
WO2020063673A1_ADC-4 payload |
Undisclosed |
WO2020063673A1_ADC-4 linker |
[7] | |
WO2020063673A1 ADC-5 |
WO2020063673A1_ADC-5 payload |
Undisclosed |
WO2020063673A1_ADC-5 linker |
[7] | |
WO2020063673A1 ADC-6 |
WO2020063673A1_ADC-6 payload |
Undisclosed |
WO2020063673A1_ADC-6 linker |
[7] | |
WO2020063673A1 ADC-7 |
WO2020063673A1_ADC-7 payload |
Undisclosed |
WO2020063673A1_ADC-7 linker |
[7] | |
WO2020063673A1 ADC-8 |
WO2020063673A1_ADC-8 payload |
Undisclosed |
WO2020063673A1_ADC-8 linker |
[7] |
Anti-CD276 mAb m276-SL
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
M276-SL-PBD |
PBD dimer |
Human Deoxyribonucleic acid (hDNA) |
Mc-Val-Ala |
[8] |
Anti-human CD276 mAb
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
B7H3-EC3 DAR4.1 |
NAMPT inhibitor 4 |
Nicotinamide phosphoribosyltransferase (NAMPT) |
Mc-Val-Ala |
[9] | |
B7H3-EC3 DAR7.8 |
NAMPT inhibitor 4 |
Nicotinamide phosphoribosyltransferase (NAMPT) |
Mc-Val-Ala |
[9] | |
B7H3-EC5 |
NAMPT inhibitor 6 |
Nicotinamide phosphoribosyltransferase (NAMPT) |
Open-chain glycine maleimide-PEG |
[9] | |
B7H3-EC4 |
NAMPT inhibitor 5 |
Nicotinamide phosphoribosyltransferase (NAMPT) |
Open-chain glycine maleimide |
[9] | |
B7H3-EC2 |
NAMPT inhibitor 6 |
Nicotinamide phosphoribosyltransferase (NAMPT) |
Maleimido-caproyl |
[9] | |
B7H3-EC1 |
NAMPT inhibitor 4 |
Nicotinamide phosphoribosyltransferase (NAMPT) |
Maleimido-caproyl |
[9] | |
CN109069633A ADC-1 |
CN109069633A ADC-1 payload |
Undisclosed |
CN109069633A ADC-1 linker |
[10] | |
CN109069633A ADC-2 |
CN109069633A ADC-2 payload |
Undisclosed |
CN109069633A ADC-2 linker |
[10] | |
CN109069633A ADC-3 |
CN109069633A ADC-3 payload |
Undisclosed |
CN109069633A ADC-3 linker |
[10] |
Antibody V3
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
CN115969996A ADC1 |
Exatecan |
DNA topoisomerase 1 (TOP1) |
CB07 linker |
[11] | |
CN115969996A ADC2 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[11] | |
CN115969996A ADC3 |
Exatecan |
DNA topoisomerase 1 (TOP1) |
CB07 linker |
[11] |
B7-H3 mAb 401
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
37235999 ADC 401-4 |
Monomethyl auristatin E |
Microtubule (MT) |
Fmoc-Val-Cit-PAB-PNP |
[12] |
B7-H3-ABBV-155
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
B7-H3-ABBV-155-L101-D101 |
Compound D101 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-ABBV-155-L102-D101 |
Compound D101 |
Undisclosed |
L102 linker |
[13] | |
B7-H3-ABBV-155-L103-D101 |
Compound D101 |
Undisclosed |
L103 linker |
[13] | |
B7-H3-ABBV-155-L101-D102 |
Compound D102 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-ABBV-155-L101-D103 |
Compound D103 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-ABBV-155-L101-D104 |
Compound D104 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-ABBV-155-L102-D102 |
Compound D102 |
Undisclosed |
L102 linker |
[13] | |
B7-H3-ABBV-155-L102-D103 |
Compound D103 |
Undisclosed |
L102 linker |
[13] | |
B7-H3-ABBV-155-L102-D104 |
Compound D104 |
Undisclosed |
L102 linker |
[13] |
B7-H3-DS-5573a
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
B7-H3-DS-5573a-L101-D101 |
Compound D101 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-DS-5573a-L102-D101 |
Compound D101 |
Undisclosed |
L102 linker |
[13] | |
B7-H3-DS-5573a-L103-D101 |
Compound D101 |
Undisclosed |
L103 linker |
[13] | |
B7-H3-DS-5573a-L101-D102 |
Compound D102 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-DS-5573a-L101-D103 |
Compound D103 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-DS-5573a-L101-D104 |
Compound D104 |
Undisclosed |
L101 linker |
[13] | |
B7-H3-DS-5573a-L102-D102 |
Compound D102 |
Undisclosed |
L102 linker |
[13] | |
B7-H3-DS-5573a-L102-D103 |
Compound D103 |
Undisclosed |
L102 linker |
[13] | |
B7-H3-DS-5573a-L102-D104 |
Compound D104 |
Undisclosed |
L102 linker |
[13] |
B7H3 antibody
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
CN115429893A ADC15 |
Undisclosed |
Undisclosed |
Undisclosed |
[14] |
B7H3 Y107 A121C
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
CN118414170A T-2-AB |
T-2 |
Undisclosed |
T-2 linker |
[15] | |
CN118414170A T-3-AB |
T-3 |
Undisclosed |
T-3 linker |
[15] | |
CN118414170A T-4-AB |
T-4 |
Undisclosed |
T-4 linker |
[15] | |
CN118414170A T-5-AB |
T-3 |
Undisclosed |
T-5 linker |
[15] | |
CN118414170A T-6-AB |
T-6 |
Undisclosed |
T-6 linker |
[15] | |
CN118414170A T-8-AB |
T-8 |
Undisclosed |
T-8 linker |
[15] | |
CN118414170A T-9-AB |
T-9 |
Undisclosed |
T-9 linker |
[15] | |
CN118414170A T-10-AB |
T-10 |
Undisclosed |
T-5 linker |
[15] | |
CN118414170A T-11-AB |
T-11 |
Undisclosed |
T-5 linker |
[15] | |
CN118414170A T-12-AB |
T-12 |
Undisclosed |
T-5 linker |
[15] | |
CN118414170A T-13-AB |
T-13 |
Undisclosed |
T-5 linker |
[15] | |
CN118414170A T-14-AB |
T-14 |
Undisclosed |
T-14 linker |
[15] | |
CN118414170A T-15-AB |
T-15 |
Undisclosed |
T-4 linker |
[15] | |
CN118414170A T-102-AB |
T-102 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-103-AB |
T-103 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-104-AB |
T-104 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-110-AB |
T-110 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-111-AB |
T-111 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-112-AB |
T-112 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-113-AB |
T-113 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-115-AB |
T-115 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-116-AB |
T-116 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-117-AB |
T-116 |
Undisclosed |
T-117 linker |
[15] | |
CN118414170A T-118-AB |
T-118 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-119-AB |
T-119 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-120-AB |
T-120 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-121-AB |
T-121 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-122-AB |
T-122 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-123-AB |
T-123 |
Undisclosed |
T-102 linker |
[15] | |
CN118414170A T-124-AB |
T-122 |
Undisclosed |
T-124 linker |
[15] | |
CN118414170A T-125-AB |
T-123 |
Undisclosed |
T-125 linker |
[15] | |
CN118414170A T-127-AB |
T-122 |
Undisclosed |
Undisclosed |
[15] | |
CN118414170A T-129-AB |
T-129 |
Undisclosed |
Undisclosed |
[15] | |
CN118414170A T-132-AB |
T-132 |
Undisclosed |
T-132 linker |
[15] | |
CN118414170A T-133-AB |
T-133 |
Undisclosed |
T-132 linker |
[15] | |
CN118414170A T-134-AB |
T-134 |
Undisclosed |
T-132 linker |
[15] | |
CN118414170A T-135-AB |
T-135 |
Undisclosed |
T-132 linker |
[15] |
B7H3-C1
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
B7H3-C1-ADC-05 (DAR4) |
B7H3-C1-ADC-05(DAR4) payload |
Undisclosed |
B7H3-C1-ADC-05(DAR4) linker |
[1] | |
B7H3-C1-ADC-07 (DAR4) |
B7H3-C1-ADC-07(DAR4) payload |
Undisclosed |
B7H3-C1-ADC-07(DAR4) linker |
[1] | |
B7H3-C1-ADC-08 (DAR4) |
B7H3-C1-ADC-08(DAR4) payload |
Undisclosed |
B7H3-C1-ADC-08(DAR4) linker |
[1] | |
B7H3-ADC-21 (DAR8) |
B7H3-ADC-21(DAR8) payload |
Undisclosed |
B7H3-ADC-21(DAR8) linker |
[1] | |
B7H3-ADC-21 (DAR2) |
B7H3-ADC-21(DAR2) payload |
Undisclosed |
B7H3-ADC-21(DAR2) linker |
[1] | |
B7H3-C1-ADC-21 (DAR4) |
B7H3-C1-ADC-21(DAR4) payload |
Undisclosed |
B7H3-C1-ADC-21(DAR4) linker |
[1] | |
B7H3-ADC-21 (DAR6) |
B7H3-ADC-21(DAR6) payload |
Undisclosed |
B7H3-ADC-21(DAR6) linker |
[1] |
chAb11
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb11-CZ |
chAb11-CZ payload |
Undisclosed |
chAb11-CZ linker |
[16] |
chAb13
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb13-CZ |
chAb13-CZ payload |
Undisclosed |
chAb13-CZ linker |
[16] |
chAb14
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb14-CZ |
chAb14-CZ payload |
Undisclosed |
chAb14-CZ linker |
[16] |
chAb16
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb16-CZ |
chAb16-CZ payload |
Undisclosed |
chAb16-CZ linker |
[16] |
chAb18
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb18-CZ |
chAb18-CZ payload |
Undisclosed |
chAb18-CZ linker |
[16] |
chAb2 (chimra IgG1)
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb2-CZ |
chAb2-CZ payload |
Undisclosed |
chAb2-CZ linker |
[16] |
chAb3
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb3-CZ |
chAb3-CZ payload |
Undisclosed |
chAb3-CZ linker |
[16] |
chAb4
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb4-CZ |
chAb4-CZ payload |
Undisclosed |
chAb4-CZ linker |
[16] |
chAb6
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChAb6-CZ |
chAb6-CZ payload |
Undisclosed |
chAb6-CZ linker |
[16] |
chmAb-A
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChmAb-A B7-H3-ADC |
Monomethyl auristatin E |
Microtubule (MT) |
Mc-Val-Cit-PABC |
[17] |
chmAb-B
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChmAb-B B7-H3-ADC |
Monomethyl auristatin E |
Microtubule (MT) |
Mc-Val-Cit-PABC |
[17] |
chmAb-C
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChmAb-C B7-H3-ADC |
Monomethyl auristatin E |
Microtubule (MT) |
Mc-Val-Cit-PABC |
[17] |
chmAb-D
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ChmAb-D B7-H3-ADC |
Monomethyl auristatin E |
Microtubule (MT) |
Mc-Val-Cit-PABC |
[17] |
Enoblituzumab
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
Enoblituzumab-ADC-24-1 |
Enoblituzumab-ADC-24-1 payload |
Undisclosed |
Enoblituzumab-ADC-24-1 linker |
[2] | |
Enoblituzumab-ADC-24-2 |
Enoblituzumab-ADC-24-2 payload |
Undisclosed |
Enoblituzumab-ADC-24-2 linker |
[2] | |
Enoblituzumab-ADC-24-3 |
Enoblituzumab-ADC-24-3 payload |
Undisclosed |
Enoblituzumab-ADC-24-3 linker |
[2] | |
Enoblituzumab-ADC-24-4 |
Enoblituzumab-ADC-24-4 payload |
Undisclosed |
Enoblituzumab-ADC-24-4 linker |
[2] | |
Enoblituzumab-ADC-24-5 |
Enoblituzumab-ADC-24-5 payload |
Undisclosed |
Enoblituzumab-ADC-24-5 linker |
[2] | |
Enoblituzumab-ADC-24-6 |
Enoblituzumab-ADC-24-6 payload |
Undisclosed |
Enoblituzumab-ADC-24-6 linker |
[2] | |
Enoblituzumab-ADC-24-7 |
Enoblituzumab-ADC-24-7 payload |
Undisclosed |
Enoblituzumab-ADC-24-7 linker |
[2] | |
Enoblituzumab-ADC-24-8 |
Enoblituzumab-ADC-24-8 payload |
Undisclosed |
Enoblituzumab-ADC-24-8 linker |
[2] | |
Enoblituzumab-ADC-24-9 |
Enoblituzumab-ADC-24-9 payload |
Undisclosed |
Enoblituzumab-ADC-24-9 linker |
[2] | |
Enoblituzumab-ADC-24-10 |
Enoblituzumab-ADC-24-10 payload |
Undisclosed |
Enoblituzumab-ADC-24-10 linker |
[2] | |
Enoblituzumab-ADC-24-11 |
Enoblituzumab-ADC-24-11 payload |
Undisclosed |
Enoblituzumab-ADC-24-11 linker |
[2] | |
Enoblituzumab-ADC-24-12 |
Enoblituzumab-ADC-24-12 payload |
Undisclosed |
Enoblituzumab-ADC-24-12 linker |
[2] | |
Enoblituzumab-ADC-24-13 |
Enoblituzumab-ADC-24-13 payload |
Undisclosed |
Enoblituzumab-ADC-24-13 linker |
[2] | |
Enoblituzumab-ADC-Tb1-1 |
Enoblituzumab-ADC-Tb1-1 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-1 linker |
[1] | |
Enoblituzumab-ADC-Tb1-2 |
Enoblituzumab-ADC-Tb1-2 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-2 linker |
[1] | |
Enoblituzumab-ADC-Tb1-3 |
Enoblituzumab-ADC-Tb1-3 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-3 linker |
[1] | |
Enoblituzumab-ADC-Tb1-4 |
Enoblituzumab-ADC-Tb1-4 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-4 linker |
[1] | |
Enoblituzumab-ADC-Tb1-5 |
Enoblituzumab-ADC-Tb1-5 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-5 linker |
[1] | |
Enoblituzumab-ADC-Tb1-6 |
Enoblituzumab-ADC-Tb1-6 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-6 linker |
[1] | |
Enoblituzumab-ADC-Tb1-7 |
Enoblituzumab-ADC-Tb1-7 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-7 linker |
[1] | |
Enoblituzumab-ADC-Tb1-8 |
Enoblituzumab-ADC-Tb1-8 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-8 linker |
[1] | |
Enoblituzumab-ADC-Tb1-9 |
Enoblituzumab-ADC-Tb1-9 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-9 linker |
[1] | |
Enoblituzumab-ADC-Tb1-10 |
Enoblituzumab-ADC-Tb1-10 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-10 linker |
[1] | |
Enoblituzumab-ADC-Tb1-11 |
Enoblituzumab-ADC-Tb1-11 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-11 linker |
[1] | |
Enoblituzumab-ADC-Tb1-12 |
Enoblituzumab-ADC-Tb1-12 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-12 linker |
[1] | |
Enoblituzumab-ADC-Tb1-13 |
Enoblituzumab-ADC-Tb1-13 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-13 linker |
[1] | |
Enoblituzumab-ADC-Tb1-14 |
Enoblituzumab-ADC-Tb1-14 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-14 linker |
[1] | |
Enoblituzumab-ADC-Tb1-15 |
Enoblituzumab-ADC-Tb1-15 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-15 linker |
[1] | |
Enoblituzumab-ADC-Tb1-16 |
Enoblituzumab-ADC-Tb1-16 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-16 linker |
[1] | |
Enoblituzumab-ADC-Tb1-17 |
Enoblituzumab-ADC-Tb1-17 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-17 linker |
[1] | |
Enoblituzumab-ADC-Tb1-18 |
Enoblituzumab-ADC-Tb1-18 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-18 linker |
[1] | |
Enoblituzumab-ADC-Tb1-19 |
Enoblituzumab-ADC-Tb1-19 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-19 linker |
[1] | |
Enoblituzumab-ADC-Tb1-20 |
Enoblituzumab-ADC-Tb1-20 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-20 linker |
[1] | |
Enoblituzumab-ADC-Tb1-21 |
Enoblituzumab-ADC-Tb1-21 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-21 linker |
[1] | |
Enoblituzumab-ADC-Tb1-22 |
Enoblituzumab-ADC-Tb1-22 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-22 linker |
[1] | |
Enoblituzumab-ADC-Tb1-23 |
Enoblituzumab-ADC-Tb1-23 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-23 linker |
[1] | |
Enoblituzumab-ADC-Tb1-24 |
Enoblituzumab-ADC-Tb1-24 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-24 linker |
[1] | |
Enoblituzumab-ADC-Tb1-25 |
Enoblituzumab-ADC-Tb1-25 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-25 linker |
[1] | |
Enoblituzumab-ADC-Tb1-26 |
Enoblituzumab-ADC-Tb1-26 payload |
Undisclosed |
Enoblituzumab-ADC-Tb1-26 linker |
[1] |
hmAb-C
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HmAb-C-DUBA |
seco-DUBA |
Human Deoxyribonucleic acid (hDNA) |
Mal-PEG2-Val-Cit-PABA-Cyclization Spacer |
[17] |
Hu276 mAb
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
CD276 mAb-MMAF |
Monomethyl auristatin F |
Microtubule (MT) |
DBM linker |
[18] | |
CD276 mAb-IMQ |
imiquimod |
Toll-like receptor 7 (TLR7); Toll-like receptor 8 (TLR8) |
Phosphine-azide |
[18] | |
CD276 mAb-MMAF/IMQ |
Monomethyl auristatin F; imiquimod |
Undisclosed |
DBM linker |
[18] |
huAb13v1
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb13v1-CZ |
huAb13v1-CZ payload |
Undisclosed |
huAb13v1-CZ linker |
[16] | |
HuAb13v1-TX |
huAb13v1-TX payload |
Undisclosed |
huAb13v1-TX linker |
[16] | |
HuAb13v1-TV |
huAb13v1-TV payload |
Undisclosed |
huAb13v1-TV linker |
[16] | |
HuAb13v1-AAA |
huAb13v1-AAA payload |
Undisclosed |
huAb13v1-AAA linker |
[16] | |
HuAb13v1-AAD |
huAb13v1-AAD payload |
Undisclosed |
huAb13v1-AAD linker |
[16] | |
HuAb13v1-WD |
huAb13v1-WD payload |
Undisclosed |
huAb13v1-WD linker |
[16] | |
HuAb13v1-LB |
huAb13v1-LB payload |
Undisclosed |
huAb13v1-LB linker |
[16] | |
HuAb13v1-ZT |
huAb13v1-ZT payload |
Undisclosed |
huAb13v1-ZT linker |
[16] | |
HuAb13v1-ZZ |
huAb13v1-ZZ payload |
Undisclosed |
huAb13v1-ZZ linker |
[16] | |
HuAb13v1-XW |
huAb13v1-XW payload |
Undisclosed |
huAb13v1-XW linker |
[16] | |
HuAb13v1-SE |
huAb13v1-SE payload |
Undisclosed |
huAb13v1-SE linker |
[16] | |
HuAb13v1-SR |
huAb13v1-SR payload |
Undisclosed |
huAb13v1-SR linker |
[16] | |
HuAb13v1-YG |
huAb13v1-YG payload |
Undisclosed |
huAb13v1-YG linker |
[16] | |
HuAb13v1-KZ |
huAb13v1-KZ payload |
Undisclosed |
huAb13v1-KZ linker |
[16] | |
HuAb13v1-WD E2 |
huAb13v1-WD E2 payload |
Undisclosed |
huAb13v1-WD E2 linker |
[16] | |
HuAb13v1-TX E2 |
huAb13v1-TX E2 payload |
Undisclosed |
huAb13v1-TX E2 linker |
[16] |
huAb18v1
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v1-CZ |
huAb18v1-CZ payload |
Undisclosed |
huAb18v1-CZ linker |
[16] |
huAb18v10
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v10-CZ |
huAb18v10-CZ payload |
Undisclosed |
huAb18v10-CZ linker |
[16] |
huAb18v2
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v2-CZ |
huAb18v2-CZ payload |
Undisclosed |
huAb18v2-CZ linker |
[16] |
huAb18v3
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v3-CZ |
huAb18v3-CZ payload |
Undisclosed |
huAb18v3-CZ linker |
[16] |
huAb18v4
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v4-CZ |
huAb18v4-CZ payload |
Undisclosed |
huAb18v4-CZ linker |
[16] |
huAb18v5
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v5-CZ |
huAb18v5-CZ payload |
Undisclosed |
huAb18v5-CZ linker |
[16] |
huAb18v6
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v6-CZ |
huAb18v6-CZ payload |
Undisclosed |
huAb18v6-CZ linker |
[16] |
huAb18v7
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v7-CZ |
huAb18v7-CZ payload |
Undisclosed |
huAb18v7-CZ linker |
[16] |
huAb18v8
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v8-CZ |
huAb18v8-CZ payload |
Undisclosed |
huAb18v8-CZ linker |
[16] |
huAb18v9
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb18v9-CZ |
huAb18v9-CZ payload |
Undisclosed |
huAb18v9-CZ linker |
[16] |
huAb3v1
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v1-CZ |
huAb3v1-CZ payload |
Undisclosed |
huAb3v1-CZ linker |
[16] |
huAb3v2
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v2-CZ |
huAb3v2-CZ payload |
Undisclosed |
huAb3v2-CZ linker |
[16] |
huAb3v2.2
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v2.2-CZ |
huAb3v2.2-CZ payload |
Undisclosed |
huAb3v2.2-CZ linker |
[16] |
huAb3v2.3
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v2.3-CZ |
huAb3v2.3-CZ payload |
Undisclosed |
huAb3v2.3-CZ linker |
[16] |
huAb3v2.5
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v2.5-CZ |
huAb3v2.5-CZ payload |
Undisclosed |
huAb3v2.5-CZ linker |
[16] | |
HuAb3v2.5-TX |
huAb3v2.5-TX payload |
Undisclosed |
huAb3v2.5-TX linker |
[16] | |
HuAb3v2.5-TV |
huAb3v2.5-TV payload |
Undisclosed |
huAb3v2.5-TV linker |
[16] | |
HuAb3v2.5-YY |
huAb3v2.5-YY payload |
Undisclosed |
huAb3v2.5-YY linker |
[16] | |
HuAb3v2.5-AAA |
huAb3v2.5-AAA payload |
Undisclosed |
huAb3v2.5-AAA linker |
[16] | |
HuAb3v2.5-AAD |
huAb3v2.5-AAD payload |
Undisclosed |
huAb3v2.5-AAD linker |
[16] | |
HuAb3v2.5-WD |
huAb3v2.5-WD payload |
Undisclosed |
huAb3v2.5-WD linker |
[16] | |
HuAb3v2.5-LB |
huAb3v2.5-LB payload |
Undisclosed |
huAb3v2.5-LB linker |
[16] | |
HuAb3v2.5-ZT |
huAb3v2.5-ZT payload |
Undisclosed |
huAb3v2.5-ZT linker |
[16] | |
HuAb3v2.5-ZZ |
huAb3v2.5-ZZ payload |
Undisclosed |
huAb3v2.5-ZZ linker |
[16] | |
HuAb3v2.5-XW |
huAb3v2.5-XW payload |
Undisclosed |
huAb3v2.5-XW linker |
[16] | |
HuAb3v2.5-SE |
huAb3v2.5-SE payload |
Undisclosed |
huAb3v2.5-SE linker |
[16] | |
HuAb3v2.5-SR |
huAb3v2.5-SR payload |
Undisclosed |
huAb3v2.5-SR linker |
[16] | |
HuAb3v2.5-YG |
huAb3v2.5-YG payload |
Undisclosed |
huAb3v2.5-YG linker |
[16] | |
HuAb3v2.5-KZ |
huAb3v2.5-KZ payload |
Undisclosed |
huAb3v2.5-KZ linker |
[16] |
huAb3v2.6
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v2.6-CZ |
huAb3v2.6-CZ payload |
Undisclosed |
huAb3v2.6-CZ linker |
[16] | |
HuAb3v2.6-TX |
huAb3v2.6-TX payload |
Undisclosed |
huAb3v2.6-TX linker |
[16] | |
HuAb3v2.6-TV |
huAb3v2.6-TV payload |
Undisclosed |
huAb3v2.6-TV linker |
[16] | |
HuAb3v2.6-YY |
huAb3v2.6-YY payload |
Undisclosed |
huAb3v2.6-YY linker |
[16] | |
HuAb3v2.6-AAA |
huAb3v2.6-AAA payload |
Undisclosed |
huAb3v2.6-AAA linker |
[16] | |
HuAb3v2.6-AAD |
huAb3v2.6-AAD payload |
Undisclosed |
huAb3v2.6-AAD linker |
[16] | |
HuAb3v2.6-WD |
huAb3v2.6-WD payload |
Undisclosed |
huAb3v2.6-WD linker |
[16] | |
HuAb3v2.6-LB |
huAb3v2.6-LB payload |
Undisclosed |
huAb3v2.6-LB linker |
[16] | |
HuAb3v2.6-ZT |
huAb3v2.6-ZT payload |
Undisclosed |
huAb3v2.6-ZT linker |
[16] | |
HuAb3v2.6-ZZ |
huAb3v2.6-ZZ payload |
Undisclosed |
huAb3v2.6-ZZ linker |
[16] | |
HuAb3v2.6-XW |
huAb3v2.6-XW payload |
Undisclosed |
huAb3v2.6-XW linker |
[16] | |
HuAb3v2.6-SE |
huAb3v2.6-SE payload |
Undisclosed |
huAb3v2.6-SE linker |
[16] | |
HuAb3v2.6-SR |
huAb3v2.6-SR payload |
Undisclosed |
huAb3v2.6-SR linker |
[16] | |
HuAb3v2.6-YG |
huAb3v2.6-YG payload |
Undisclosed |
huAb3v2.6-YG linker |
[16] | |
HuAb3v2.6-KZ |
huAb3v2.6-KZ payload |
Undisclosed |
huAb3v2.6-KZ linker |
[16] |
huAb3v2.8
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v2.8-CZ |
huAb3v2.8-CZ payload |
Undisclosed |
huAb3v2.8-CZ linker |
[16] |
huAb3v2.9
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v2.9-CZ |
huAb3v2.9-CZ payload |
Undisclosed |
huAb3v2.9-CZ linker |
[16] | |
HuAb3v2.9-TX |
huAb3v2.9-TX payload |
Undisclosed |
huAb3v2.9-TX linker |
[16] |
huAb3v3
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v3-CZ |
huAb3v3-CZ payload |
Undisclosed |
huAb3v3-CZ linker |
[16] |
huAb3v4
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v4-CZ |
huAb3v4-CZ payload |
Undisclosed |
huAb3v4-CZ linker |
[16] |
huAb3v5
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v5-CZ |
huAb3v5-CZ payload |
Undisclosed |
huAb3v5-CZ linker |
[16] |
huAb3v6
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
HuAb3v6-CZ |
huAb3v6-CZ payload |
Undisclosed |
huAb3v6-CZ linker |
[16] |
Ifinatamab
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ZA202500415A-ADC Example 4 |
NMT inhibitor 1 |
N-Myristoyltransferase (NMT) |
ZA202500415A-ADC-Example-1-Linker |
[19] | |
SG11202408662TA ADC-C1 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[20] | |
SG11202408662TA ADC-C2 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C3 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C4 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C5 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C6 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C7 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C8 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C9 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C10 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C11 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C12 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C13 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
SG11202408662TA ADC-C14 |
Undisclosed |
Undisclosed |
Undisclosed |
[20] | |
WO2024165045A1 ADC-B |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-4 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-5 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-6 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-7 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-8 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-9 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-10 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-11 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-12 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-13 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-14 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
WO2024165045A1 ADC-16 |
Undisclosed |
Undisclosed |
Undisclosed |
[21] | |
CN119317630A ADC-C1 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[22] | |
CN119317630A ADC-C2 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[22] | |
CN119317630A ADC-C3 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C3 Linker |
[22] | |
CN119317630A ADC-C4 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C3 Linker |
[22] | |
CN119317630A ADC-C5 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C5 Linker |
[22] | |
CN119317630A ADC-C6 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C5 Linker |
[22] | |
CN119317630A ADC-C7 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C7 Linker |
[22] | |
CN119317630A ADC-C8 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C8 Linker |
[22] | |
CN119317630A ADC-C9 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C9 Linker |
[22] | |
CN119317630A ADC-C10 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C10 Linker |
[22] | |
CN119317630A ADC-C11 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C11 Linker |
[22] | |
CN119317630A ADC-C12 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C12 Linker |
[22] | |
CN119317630A ADC-C13 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C13 Linker |
[22] | |
CN119317630A ADC-C14 |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
CN119317630A ADC-C14 Linker |
[22] |
Mirzotamab
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
Mirzotamab-ADC-Tb1-1 |
Mirzotamab-ADC-Tb1-1 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-1 linker |
[1] | |
Mirzotamab-ADC-Tb1-2 |
Mirzotamab-ADC-Tb1-2 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-2 linker |
[1] | |
Mirzotamab-ADC-Tb1-3 |
Mirzotamab-ADC-Tb1-3 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-3 linker |
[1] | |
Mirzotamab-ADC-Tb1-4 |
Mirzotamab-ADC-Tb1-4 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-4 linker |
[1] | |
Mirzotamab-ADC-Tb1-5 |
Mirzotamab-ADC-Tb1-5 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-5 linker |
[1] | |
Mirzotamab-ADC-Tb1-6 |
Mirzotamab-ADC-Tb1-6 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-6 linker |
[1] | |
Mirzotamab-ADC-Tb1-7 |
Mirzotamab-ADC-Tb1-7 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-7 linker |
[1] | |
Mirzotamab-ADC-Tb1-8 |
Mirzotamab-ADC-Tb1-8 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-8 linker |
[1] | |
Mirzotamab-ADC-Tb1-9 |
Mirzotamab-ADC-Tb1-9 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-9 linker |
[1] | |
Mirzotamab-ADC-Tb1-10 |
Mirzotamab-ADC-Tb1-10 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-10 linker |
[1] | |
Mirzotamab-ADC-Tb1-11 |
Mirzotamab-ADC-Tb1-11 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-11 linker |
[1] | |
Mirzotamab-ADC-Tb1-12 |
Mirzotamab-ADC-Tb1-12 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-12 linker |
[1] | |
Mirzotamab-ADC-Tb1-13 |
Mirzotamab-ADC-Tb1-13 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-13 linker |
[1] | |
Mirzotamab-ADC-Tb1-14 |
Mirzotamab-ADC-Tb1-14 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-14 linker |
[1] | |
Mirzotamab-ADC-Tb1-15 |
Mirzotamab-ADC-Tb1-15 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-15 linker |
[1] | |
Mirzotamab-ADC-Tb1-16 |
Mirzotamab-ADC-Tb1-16 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-16 linker |
[1] | |
Mirzotamab-ADC-Tb1-17 |
Mirzotamab-ADC-Tb1-17 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-17 linker |
[1] | |
Mirzotamab-ADC-Tb1-18 |
Mirzotamab-ADC-Tb1-18 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-18 linker |
[1] | |
Mirzotamab-ADC-Tb1-19 |
Mirzotamab-ADC-Tb1-19 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-19 linker |
[1] | |
Mirzotamab-ADC-Tb1-20 |
Mirzotamab-ADC-Tb1-20 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-20 linker |
[1] | |
Mirzotamab-ADC-Tb1-21 |
Mirzotamab-ADC-Tb1-21 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-21 linker |
[1] | |
Mirzotamab-ADC-Tb1-22 |
Mirzotamab-ADC-Tb1-22 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-22 linker |
[1] | |
Mirzotamab-ADC-Tb1-23 |
Mirzotamab-ADC-Tb1-23 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-23 linker |
[1] | |
Mirzotamab-ADC-Tb1-24 |
Mirzotamab-ADC-Tb1-24 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-24 linker |
[1] | |
Mirzotamab-ADC-Tb1-25 |
Mirzotamab-ADC-Tb1-25 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-25 linker |
[1] | |
Mirzotamab-ADC-Tb1-26 |
Mirzotamab-ADC-Tb1-26 payload |
Undisclosed |
Mirzotamab-ADC-Tb1-26 linker |
[1] |
Non-pH-B7-H3 Ab
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
Non-pH-B7-H3 Ab-Dxd |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[23] | |
Non-pH-B7-H3 Ab-MMAE |
Monomethyl auristatin E |
Microtubule (MT) |
Mc-Val-Cit-PABC |
[23] |
Omburtamab
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
Omburtamab-ADC-Tb1-1 |
Omburtamab-ADC-Tb1-1 payload |
Undisclosed |
Omburtamab-ADC-Tb1-1 linker |
[1] | |
Omburtamab-ADC-Tb1-2 |
Omburtamab-ADC-Tb1-2 payload |
Undisclosed |
Omburtamab-ADC-Tb1-2 linker |
[1] | |
Omburtamab-ADC-Tb1-3 |
Omburtamab-ADC-Tb1-3 payload |
Undisclosed |
Omburtamab-ADC-Tb1-3 linker |
[1] | |
Omburtamab-ADC-Tb1-4 |
Omburtamab-ADC-Tb1-4 payload |
Undisclosed |
Omburtamab-ADC-Tb1-4 linker |
[1] | |
Omburtamab-ADC-Tb1-5 |
Omburtamab-ADC-Tb1-5 payload |
Undisclosed |
Omburtamab-ADC-Tb1-5 linker |
[1] | |
Omburtamab-ADC-Tb1-6 |
Omburtamab-ADC-Tb1-6 payload |
Undisclosed |
Omburtamab-ADC-Tb1-6 linker |
[1] | |
Omburtamab-ADC-Tb1-7 |
Omburtamab-ADC-Tb1-7 payload |
Undisclosed |
Omburtamab-ADC-Tb1-7 linker |
[1] | |
Omburtamab-ADC-Tb1-8 |
Omburtamab-ADC-Tb1-8 payload |
Undisclosed |
Omburtamab-ADC-Tb1-8 linker |
[1] | |
Omburtamab-ADC-Tb1-9 |
Omburtamab-ADC-Tb1-9 payload |
Undisclosed |
Omburtamab-ADC-Tb1-9 linker |
[1] | |
Omburtamab-ADC-Tb1-10 |
Omburtamab-ADC-Tb1-10 payload |
Undisclosed |
Omburtamab-ADC-Tb1-10 linker |
[1] | |
Omburtamab-ADC-Tb1-11 |
Omburtamab-ADC-Tb1-11 payload |
Undisclosed |
Omburtamab-ADC-Tb1-11 linker |
[1] | |
Omburtamab-ADC-Tb1-12 |
Omburtamab-ADC-Tb1-12 payload |
Undisclosed |
Omburtamab-ADC-Tb1-12 linker |
[1] | |
Omburtamab-ADC-Tb1-13 |
Omburtamab-ADC-Tb1-13 payload |
Undisclosed |
Omburtamab-ADC-Tb1-13 linker |
[1] | |
Omburtamab-ADC-Tb1-14 |
Omburtamab-ADC-Tb1-14 payload |
Undisclosed |
Omburtamab-ADC-Tb1-14 linker |
[1] | |
Omburtamab-ADC-Tb1-15 |
Omburtamab-ADC-Tb1-15 payload |
Undisclosed |
Omburtamab-ADC-Tb1-15 linker |
[1] | |
Omburtamab-ADC-Tb1-16 |
Omburtamab-ADC-Tb1-16 payload |
Undisclosed |
Omburtamab-ADC-Tb1-16 linker |
[1] | |
Omburtamab-ADC-Tb1-17 |
Omburtamab-ADC-Tb1-17 payload |
Undisclosed |
Omburtamab-ADC-Tb1-17 linker |
[1] | |
Omburtamab-ADC-Tb1-18 |
Omburtamab-ADC-Tb1-18 payload |
Undisclosed |
Omburtamab-ADC-Tb1-18 linker |
[1] | |
Omburtamab-ADC-Tb1-19 |
Omburtamab-ADC-Tb1-19 payload |
Undisclosed |
Omburtamab-ADC-Tb1-19 linker |
[1] | |
Omburtamab-ADC-Tb1-20 |
Omburtamab-ADC-Tb1-20 payload |
Undisclosed |
Omburtamab-ADC-Tb1-20 linker |
[1] | |
Omburtamab-ADC-Tb1-21 |
Omburtamab-ADC-Tb1-21 payload |
Undisclosed |
Omburtamab-ADC-Tb1-21 linker |
[1] | |
Omburtamab-ADC-Tb1-22 |
Omburtamab-ADC-Tb1-22 payload |
Undisclosed |
Omburtamab-ADC-Tb1-22 linker |
[1] | |
Omburtamab-ADC-Tb1-23 |
Omburtamab-ADC-Tb1-23 payload |
Undisclosed |
Omburtamab-ADC-Tb1-23 linker |
[1] | |
Omburtamab-ADC-Tb1-24 |
Omburtamab-ADC-Tb1-24 payload |
Undisclosed |
Omburtamab-ADC-Tb1-24 linker |
[1] | |
Omburtamab-ADC-Tb1-25 |
Omburtamab-ADC-Tb1-25 payload |
Undisclosed |
Omburtamab-ADC-Tb1-25 linker |
[1] | |
Omburtamab-ADC-Tb1-26 |
Omburtamab-ADC-Tb1-26 payload |
Undisclosed |
Omburtamab-ADC-Tb1-26 linker |
[1] |
pH-B7-H3 Ab
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
pH-B7-H3 Ab-Dxd |
DX-8951 derivative (DXd) |
DNA topoisomerase 1 (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[23] | |
pH-B7-H3 Ab-MMAE |
Monomethyl auristatin E |
Microtubule (MT) |
Mc-Val-Cit-PABC |
[23] |
TPP-8567
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
Anti-B7H3 APDC 3f |
Kinesin spindle protein (KSP) inhibitor 3f |
Kinesin-like protein KIF11 (KIF11) |
Open-chain glycine maleimide |
[24] | |
Anti-B7H3 APDC 3g |
Kinesin spindle protein (KSP) inhibitor 3g |
Kinesin-like protein KIF11 (KIF11) |
Open-chain glycine maleimide |
[24] |
Undisclosed
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
IBI-129 |
Undisclosed |
Undisclosed |
Undisclosed |
||
YBL-015 |
Undisclosed |
Undisclosed |
Undisclosed |
[25] | |
64Cu-DOTAGA-alphaCD276 mAb |
Undisclosed |
Undisclosed |
Undisclosed |
[26] | |
B7-H3 ADC (Jiangsu hengrui) |
Undisclosed |
Undisclosed |
Undisclosed |
[27] | |
BVD-CD276 |
Undisclosed |
Undisclosed |
Undisclosed |
[28] | |
B7H3-MMAE |
Monomethyl auristatin E |
Microtubule (MT) |
Undisclosed |
[29] | |
NV106 |
Panobinostat |
Histone deacetylase 1 (HDAC1) |
Undisclosed |
[30] | |
NV104 |
Irinotecan |
DNA topoisomerase 1 (TOP1) |
Undisclosed |
[30] | |
NV105 |
Temozolomide |
Human Deoxyribonucleic acid (hDNA) |
Undisclosed |
[30] |
undisclosed
| ADC Info | ADC Name | Payload | Target | Linker | Ref |
|---|---|---|---|---|---|
ITC-6102RO |
Benzodiazepine dimer derivative |
Undisclosed |
Maleimide-containing OHPAS linker |
[31] | |
GLR1061 |
Undisclosed |
Undisclosed |
Undisclosed |
[32] | |
antiB7H3 MF6 |
MF6 |
Undisclosed |
Undisclosed |
[33] | |
IL317340A-1 |
TW202500135A-1 payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-2 1 |
TW202500135A-1 payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-3 |
Undisclosed |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-4 |
IL317340A-4payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-5 |
IL317340A-5payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-6 |
IL317340A-6payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-7 |
IL317340A-7payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-8 |
Topo1 inhibitor F |
DNA topoisomerase I (TOP1) |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-9 |
IL317340A-9payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-10 |
IL317340A-10payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-11 |
Undisclosed |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-12 |
Undisclosed |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-13 |
TW202500135A-1 payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
IL317340A-14 |
TW202500135A-1 payload |
Undisclosed |
Mc-Gly-Gly-Phe-Gly |
[34] | |
Production of the antibody-drug conjugate (4) |
undisclosed |
Undisclosed |
Undisclosed |
[35] |
References
