General Information of This Antigen
Antigen ID
TAR0GIFMP
Antigen Name
G-protein coupled receptor 20 (GPR20)
Gene Name
GPR20
Gene ID
2843
Sequence
MPSVSPAGPSAGAVPNATAVTTVRTNASGLEVPLFHLFARLDEELHGTFPGLWLALMAVH
GAIFLAGLVLNGLALYVFCCRTRAKTPSVIYTINLVVTDLLVGLSLPTRFAVYYGARGCL
RCAFPHVLGYFLNMHCSILFLTCICVDRYLAIVRPEGSRRCRQPACARAVCAFVWLAAGA
VTLSVLGVTGSRPCCRVFALTVLEFLLPLLVISVFTGRIMCALSRPGLLHQGRQRRVRAM
QLLLTVLIIFLVCFTPFHARQVAVALWPDMPHHTSLVVYHVAVTLSSLNSCMDPIVYCFV
TSGFQATVRGLFGQHGEREPSSGDVVSMHRSSKGSGRHHILSAGPHALTQALANGPEA

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Family
G-protein coupled receptor 1 family
Function
Orphan receptor with constitutive G(i) signaling activity that activate cyclic AMP.

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Uniprot Entry
GPR20_HUMAN
HGNC ID
HGNC:4475
KEGG ID
hsa:2843
Each Antibody-drug Conjuate AND It's Component Related to This Antigen
Full List of The ADC Related to This Antigen
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-1
WO2018135501A1_ADC-1 payload
Undisclosed
WO2018135501A1_ADC-1 linker
[1]
WO2018135501A1 ADC-2
WO2018135501A1_ADC-2 payload
Undisclosed
WO2018135501A1_ADC-2 linker
[1]
Anti-GPR20 antibody
ADC Info ADC Name Payload Target Linker Ref
DS-6157
DXd
DNA topoisomerase 1 (TOP1)
Mc-Gly-Gly-Phe-Gly
h046-H10/L1
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-11
WO2018135501A1_ADC-11 payload
Undisclosed
WO2018135501A1_ADC-11 linker
[1]
h046-H10/L6
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-12
WO2018135501A1_ADC-12 payload
Undisclosed
WO2018135501A1_ADC-12 linker
[1]
h046-H4b/L7
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-3
WO2018135501A1_ADC-3 payload
Undisclosed
WO2018135501A1_ADC-3 linker
[1]
WO2018135501A1 ADC-4
WO2018135501A1_ADC-4 payload
Undisclosed
WO2018135501A1_ADC-4 linker
[1]
WO2018135501A1 ADC-7
WO2018135501A1_ADC-7 payload
Undisclosed
WO2018135501A1_ADC-7 linker
[1]
h046-H4e/L7
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-13
WO2018135501A1_ADC-13 payload
Undisclosed
WO2018135501A1_ADC-13 linker
[1]
WO2018135501A1 ADC-14
WO2018135501A1_ADC-14 payload
Undisclosed
WO2018135501A1_ADC-14 linker
[1]
h046-H5b/L2
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-5
WO2018135501A1_ADC-5 payload
Undisclosed
WO2018135501A1_ADC-5 linker
[1]
WO2018135501A1 ADC-8
WO2018135501A1_ADC-8 payload
Undisclosed
WO2018135501A1_ADC-8 linker
[1]
h046-H8/L1
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-10
WO2018135501A1_ADC-10 payload
Undisclosed
WO2018135501A1_ADC-10 linker
[1]
h046-Hwt/L6
ADC Info ADC Name Payload Target Linker Ref
WO2018135501A1 ADC-6
WO2018135501A1_ADC-6 payload
Undisclosed
WO2018135501A1_ADC-6 linker
[1]
WO2018135501A1 ADC-9
WO2018135501A1_ADC-9 payload
Undisclosed
WO2018135501A1_ADC-9 linker
[1]
undisclosed
ADC Info ADC Name Payload Target Linker Ref
Production of the antibody-drug conjugate (5)
undisclosed
Undisclosed
Undisclosed
[2]
References
Ref 1 Anti-gpr20 antibody and anti-gpr20 antibody-drug conjugate; 2018-07-26.
Ref 2 Combination of antibody-drug conjugate with anti-SIRPα antibody