General Information of This Antigen
Antigen ID
TAR0HELFC
Antigen Name
Delta-like protein 3 (DLL3)
Gene Name
DLL3
Gene ID
10683
Synonym
Drosophila Delta homolog 3
Sequence
MVSPRMSGLLSQTVILALIFLPQTRPAGVFELQIHSFGPGPGPGAPRSPCSARLPCRLFF
RVCLKPGLSEEAAESPCALGAALSARGPVYTEQPGAPAPDLPLPDGLLQVPFRDAWPGTF
SFIIETWREELGDQIGGPAWSLLARVAGRRRLAAGGPWARDIQRAGAWELRFSYRARCEP
PAVGTACTRLCRPRSAPSRCGPGLRPCAPLEDECEAPLVCRAGCSPEHGFCEQPGECRCL
EGWTGPLCTVPVSTSSCLSPRGPSSATTGCLVPGPGPCDGNPCANGGSCSETPRSFECTC
PRGFYGLRCEVSGVTCADGPCFNGGLCVGGADPDSAYICHCPPGFQGSNCEKRVDRCSLQ
PCRNGGLCLDLGHALRCRCRAGFAGPRCEHDLDDCAGRACANGGTCVEGGGAHRCSCALG
FGGRDCRERADPCAARPCAHGGRCYAHFSGLVCACAPGYMGARCEFPVHPDGASALPAAP
PGLRPGDPQRYLLPPALGLLVAAGVAGAALLLVHVRRRGHSQDAGSRLLAGTPEPSVHAL
PDALNNLRTQEGSGDGPSSSVDWNRPEDVDPQGIYVISAPSIYAREVATPLFPPLHTGRA
GQRQHLLFPYPSSILSVK

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Function
Inhibits primary neurogenesis. May be required to divert neurons along a specific differentiation pathway. Plays a role in the formation of somite boundaries during segmentation of the paraxial mesoderm.

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Uniprot Entry
DLL3_HUMAN
HGNC ID
HGNC:2909
KEGG ID
hsa:10683
Each Antibody-drug Conjuate AND It's Component Related to This Antigen
Full List of The ADC Related to This Antigen
ADC Info ADC Name Payload Target Linker Ref
JP7560255B2 ControlADC52
Undisclosed
Undisclosed
Undisclosed
[1]
Anti-DLL3 antibody
ADC Info ADC Name Payload Target Linker Ref
SYS6040
Undisclosed
Undisclosed
A cleavable linker
FZ-AD005
DXd
DNA topoisomerase 1 (TOP1)
Mc-Val-Ala-PABC double self-immolative linker
Anti-DLL3 mAb
ADC Info ADC Name Payload Target Linker Ref
BL-M14D1
Ed-04
DNA topoisomerase 1 (TOP1)
Gly-Mal-Gly-Gly-Phe-Gly
[2]
IBI3009
NT1
DNA topoisomerase 1 (TOP1)
Undisclosed
Antibody of AMG595
ADC Info ADC Name Payload Target Linker Ref
JP7623413B2 ExampleADC61
Undisclosed
Undisclosed
Undisclosed
[3]
Glimatamab
ADC Info ADC Name Payload Target Linker Ref
JP7560255B2 ControlADC55
Undisclosed
Undisclosed
Undisclosed
[1]
Rovalpituzumab
ADC Info ADC Name Payload Target Linker Ref
Rovalpituzumab tesirine
SG3199 (SC-DR002)
Human deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala-PABC
SC-002
SG3199 (SC-DR002)
Human deoxyribonucleic acid (hDNA)
Val-Ala dipeptide linker
ADC Info ADC Name Payload Target Linker Ref
SC16.10-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.10-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.10-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.10-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.10-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.101-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.101-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.101-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.101-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.101-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.103-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.103-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.103-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.103-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.103-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.104-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.104-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.104-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.104-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.104-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.105-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.105-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.105-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.105-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.105-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.106-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.106-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.106-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.106-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.106-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.107-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.107-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.107-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.107-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.107-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.108-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.108-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.108-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.108-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.108-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.109-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.109-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.109-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.109-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.109-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.11-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.11-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.11-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.11-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.11-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.110-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.110-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.110-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.110-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.110-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.111-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.111-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.111-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.111-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.111-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.113-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.113-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.113-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.113-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.113-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.114-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.114-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.114-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.114-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.114-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.115-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.115-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.115-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.115-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.115-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.116-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.116-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.116-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.116-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.116-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.117-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.117-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.117-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.117-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.117-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.118-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.118-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.118-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.118-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.118-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.120-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.120-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.120-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.120-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.120-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.121-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.121-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.121-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.121-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.121-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.122-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.122-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.122-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.122-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.122-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.123-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.123-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.123-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.123-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.123-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.124-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.124-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.124-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.124-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.124-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.125-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.125-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.125-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.125-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.125-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.126-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.126-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.126-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.126-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.126-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.129-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.129-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.129-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.129-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.129-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.13-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.13-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.13-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.13-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.13-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.130-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.130-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.130-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.130-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.130-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.131-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.131-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.131-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.131-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.131-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.132-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.132-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.132-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.132-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.132-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.133-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.133-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.133-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.133-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.133-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.134-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.134-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.134-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.134-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.134-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.135-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.135-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.135-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.135-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.135-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.136-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.136-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.136-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.136-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.136-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.137-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.137-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.137-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.137-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.137-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.138-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.138-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.138-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.138-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.138-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.139-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.139-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.139-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.139-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.139-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.140-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.140-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.140-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.140-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.140-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.141-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.141-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.141-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.141-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.141-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.142-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.142-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.142-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.142-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.142-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.143-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.143-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.143-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.143-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.143-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.144-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.144-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.144-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.144-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.144-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.147-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.147-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.147-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.147-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.147-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.148-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.148-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.148-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.148-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.148-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.149-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.149-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.149-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.149-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.149-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.15-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.15-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.15-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.15-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.15-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.150-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.150-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.150-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.150-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.150-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.18-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.18-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.18-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.18-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.18-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.19-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.19-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.19-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.19-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.19-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.20-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.20-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.20-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.20-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.20-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.21-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.21-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.21-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.21-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.21-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.22-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.22-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.22-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.22-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.22-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.23-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.23-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.23-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.23-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.23-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.25-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.25-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.25-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.25-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.25-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.26-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.26-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.26-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.26-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.26-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.29-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.29-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.29-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.29-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.29-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.3-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.3-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.3-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.3-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.3-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.30-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.30-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.30-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.30-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.30-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.31-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.31-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.31-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.31-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.31-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.34-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.34-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.34-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.34-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.34-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.35-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.35-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.35-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.35-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.35-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.36-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.36-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.36-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.36-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.36-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.38-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.38-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.38-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.38-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.38-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.4-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.4-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.4-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.4-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.4-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.41-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.41-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.41-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.41-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.41-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.42-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.42-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.42-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.42-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.42-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.45-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.45-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.45-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.45-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.45-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.47-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.47-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.47-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.47-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.47-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.49-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.49-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.49-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.49-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.49-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.5-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.5-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.5-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.5-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.5-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.50-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.50-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.50-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.50-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.50-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.52-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.52-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.52-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.52-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.52-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.55-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.55-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.55-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.55-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.55-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.56-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.56-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.56-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.56-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.56-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.57-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.57-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.57-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.57-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.57-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.58-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.58-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.58-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.58-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.58-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.61-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.61-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.61-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.61-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.61-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.62-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.62-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.62-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.62-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.62-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.63-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.63-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.63-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.63-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.63-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.65-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.65-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.65-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.65-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.65-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.67-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.67-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.67-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.67-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.67-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.68-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.68-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.68-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.68-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.68-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.7-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.7-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.7-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.7-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.7-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.72-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.72-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.72-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.72-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.72-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.73-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.73-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.73-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.73-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.73-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.78-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.78-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.78-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.78-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.78-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.79-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.79-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.79-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.79-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.79-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.8-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.8-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.8-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.8-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.8-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.80-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.80-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.80-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.80-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.80-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.81-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.81-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.81-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.81-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.81-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.84-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.84-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.84-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.84-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.84-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SC16.88-DL1
SG2000 derivative PBD 1
Microtubule (MT)
Mal-PEG8-Val-Ala
[4]
SC16.88-DL2
SG3312
Human Deoxyribonucleic acid (hDNA)
Mc-Val-Ala
[4]
SC16.88-DL3
SG2000 derivative PBD 3
Human Deoxyribonucleic acid (hDNA)
Mal-PEG8-Val-Ala
[4]
SC16.88-DL4
SG2219
Human Deoxyribonucleic acid (hDNA)
Iodoacetamide-PEG4-Val-Ala-PABC
[4]
SC16.88-DL5
SG3199
Human Deoxyribonucleic acid (hDNA)
Mc-PEG8-Val-Ala-PABC
[4]
ADC Info ADC Name Payload Target Linker Ref
SHR-4849
SHR9265
DNA topoisomerase 1 (TOP1)
Mc-Gly-Gly-Phe-Gly
SYM004 (anti-DLL3)
ADC Info ADC Name Payload Target Linker Ref
WO2024169913A1 ADC04-01-8
B19
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
Mc-Val-Cit-PABC
[5]
WO2024169913A1 ADC04-02-8
B19
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
Mc-Val-Cit-PABC
[5]
WO2024169913A1 ADC04-06-8
B19
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
Mc-Val-Ala-PABC
[5]
WO2024169913A1 ADC04-06-4
B63
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
Mc-Val-Ala-PABC
[5]
WO2024169913A1 ADC04-07-8
B63
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
Mc-Val-Ala-PABC
[5]
WO2024169913A1 ADC04-07-4
B19
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
(Linker-02)MC-PEG-VA-PAB
[5]
WO2024169913A1 ADC04-08-8
B19
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
(Linker-02)MC-PEG-VA-PAB
[5]
WO2024169913A1 ADC04-08-4
B19
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
(Linker-03)SMCC-TAZ-PEG-VC-PAB
[5]
WO2024169913A1 ADC04-09-8
Smol006
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
Mc-Val-Cit-PABC
[5]
WO2024169913A1 ADC04-09-4
Smol006
Eukaryotic peptide chain release factor GTP-binding subunit ERF3A (GSPT1)
Mc-Val-Cit-PABC
[5]
Zocilurtatug
ADC Info ADC Name Payload Target Linker Ref
Zocilurtatug pelitecan
YL0010014
DNA topoisomerase 1 (TOP1)
VK*G-NHCH2-O linker
[6]
Undisclosed
ADC Info ADC Name Payload Target Linker Ref
ZL-1310
YL0010014
DNA topoisomerase I (TOP1)
Tumor microenviroment activable tripeptide linker
[7]
Anti-DLL3 ADC (IntoCell/Y-Biologics)
Undisclosed
Undisclosed
Undisclosed
[8]
undisclosed
ADC Info ADC Name Payload Target Linker Ref
PLB-001
Exatecan
DNA topoisomerase 1 (TOP1)
Undisclosed
[9]
WO2024043319A1 80
Undisclosed
Undisclosed
Undisclosed
[10]
CN119630431A ADC-92
CN119630431A-ADC-82-PAYLOAD
Undisclosed
CN119630431A-ADC-82-LINKER
[11]
References
Ref 1 Pharmaceuticals containing antibody-drug complexes containing hemiasterin derivatives
Ref 2 Biokin pharma Prospectus; 2022
Ref 3 Antibody-drug complexes containing hemiasterlin derivatives
Ref 4 Novel antibody conjugates and uses thereof; 2014-08-28.
Ref 5 Domide molecular glue derivative and use thereof
Ref 6 Zai lab announces strategic partnership and global license agreement with medilink therapeutics for a next generation antibody-drug conjugate program in oncology
Ref 7 A Study of ZL-1310 in Subjects With Small Cell Lung Cancer
Ref 8 Introduction to basic information on anti-DLL3 ADC (IntoCell/Y-Biologics).
Ref 9 PLB-001, a novel anti-dll3 ADC with topoisomerase 1 inhibitor-based linker-payload for treatment of SCLC
Ref 10 Antibody-drug complexes
Ref 11 Antibody-drug conjugates