General Information of This Antibody-drug Conjugate (ADC)
ADC ID
DRG0MHAHZ
ADC Name
Coltuximab ravtansine
Synonyms
Anti-CD19 humanized monoclonal antibody conjugated to DM4; Anti-CD19-DM4 immunoconjugate; Coltuximab ravtansine; HUB4-DM4, SAR34 19; HuB4-DM4; Maytansin-loaded anti-CD19 mAb; SAR-3419; SAR3419
   Click to Show/Hide
Organization
ImmunoGen, Inc.; Sanofi
Drug Status
Phase 2 (Terminated)
Indication
In total 3 Indication(s)
Acute lymphoblastic leukemia
Phase 2
Clinical Trial
Diffuse large B-cell lymphoma
Phase 2
Clinical Trial
Unspecific non-hodgkin lymphoma
Phase 1
Clinical Trial
Drug-to-Antibody Ratio
3 to 4
Structure
Antibody Name
Coltuximab
 Antibody Info 
Antigen Name
B-lymphocyte antigen CD19 (CD19)
 Antigen Info 
Payload Name
Mertansine DM4
 Payload Info 
Therapeutic Target
Microtubule (MT)
 Target Info 
Linker Name
N-succinimidyl 4-(2-pyridyldithio) butanoate (SPDB)
 Linker Info 
Conjugate Type
Random Cysteines
Combination Type
ravtansine
Puchem SID
472408086 , 223370395 , 160682393 , 404770208
Drugbank ID
DB06342
DrugMap ID
DMSGFOY
TTD ID
D00UNK
ChEBI ID
CHEMBL2109286