General Information of This Antibody-drug Conjugate (ADC)
ADC ID
DRG0HISTV
ADC Name
AVE-9633
Synonyms
AVE 9633; AVE-9633; AVE96 33; AVE9633; Anti-CD33 TAP; Anti-CD33-DM4 immunoconjugate; IMGN-633; huMY96DM4; huMy9-6-DM4
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Organization
ImmunoGen, Inc.; Sanofi
Drug Status
Phase 1 (Terminated)
Indication
In total 1 Indication(s)
Acute myeloid leukaemia
Phase 1
Clinical Trial
Drug-to-Antibody Ratio
3.5
Structure
Antibody Name
Anti-CD33 mAb huMy9-6
 Antibody Info 
Antigen Name
Myeloid cell surface antigen CD33 (CD33)
 Antigen Info 
Payload Name
Mertansine DM4
 Payload Info 
Therapeutic Target
Microtubule (MT)
 Target Info 
Linker Name
N-succinimidyl 4-(2-pyridyldithio) butanoate (SPDB)
 Linker Info 
Conjugate Type
Undisclosed
Combination Type
ravtansine
Puchem SID
160703912 , 135303445
Drugbank ID
DB06318
ChEBI ID
CHEMBL2109266