General Information of This Payload
Payload ID
PAY0LUPMV
Name
T-651 similar fusion inhibitor
Synonyms
T-651 similar fusion inhibitor
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Target(s) Envelope glycoprotein gp160 (env)
The activity data of This Payload
Standard Type Value Units Cell line Disease Model Cell line ID Reference
Half Maximal Inhibitory Concentration (IC50) 10.0±2.1 ng/mL
C597-8-H0 virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 10.2±2.7 ng/mL
93TH6.9 virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 10.5±0.8 ng/mL
SF162 virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 3.1±2.2 ng/mL
NLBal virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 42.1±4.5 ng/mL
NL4-3 virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 5.8±1.2 ng/mL
JRFL virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 6.2±0.8 ng/mL
CS81-69-E09 virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 6.3±0.6 ng/mL
CS81-4-G0 virus
Human immunodeficiency virus type 1
Undisclosed [1]
Half Maximal Inhibitory Concentration (IC50) 7.5±2.5 ng/mL
HXB2 virus
Human immunodeficiency virus type 1
Undisclosed [1]
Each Antibody-drug Conjugate Related to This Payload
References
Ref 1 CD4-BFFI: a novel, bifunctional HIV-1 entry inhibitor with high and broad antiviral potency. Antiviral Res. 2009 Sep;83(3):257-66.

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